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Musilek, Kamil
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Scholarly & Creative Works
selected scholarly works & creative activities
Article
2022
Charged pyridinium oximes with thiocarboxamide moiety are equally or less effective reactivators of organophosphate-inhibited cholinesterases compared to analogous carboxamides
Full Text via DOI:
10.1080/14756366.2022.2041628
Web of Science:
000759901800001
2022
Novel D
2
/5-HT receptor modulators related to cariprazine with potential implication to schizophrenia treatment
.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
. 232.
Full Text via DOI:
10.1016/j.ejmech.2022.114193
2021
Synthesis and In Vitro Evaluation of Novel Dopamine Receptor D
2
3,4-dihydroquinolin-2(1
H
)-one Derivatives Related to Aripiprazole
Full Text via DOI:
10.3390/biom11091262
Web of Science:
000699332600001
2021
(±)-BIGI-3h: Pentatarget-Directed Ligand combining Cholinesterase, Monoamine Oxidase, and Glycogen Synthase Kinase 3β Inhibition with Calcium Channel Antagonism and Antiaggregating Properties for Alzheimer's Disease
.
ACS CHEMICAL NEUROSCIENCE
. 12:1328-1342.
Full Text via DOI:
10.1021/acschemneuro.0c00803
Web of Science:
000643598600005
2021
Biomarkers of deoxynivalenol (DON) and its modified form DON-3-glucoside (DON-3G) in humans
Full Text via DOI:
10.1016/j.tifs.2021.02.038
Web of Science:
000632854800007
2021
Determination of K869, a Novel Oxime Reactivator of Acetylcholinesterase, in Rat Body Fluids and Tissues by Liquid-Chromatography Methods: Pharmacokinetic Study
Full Text via DOI:
10.1016/j.xphs.2021.01.031
Web of Science:
000631863100040
2021
Effects of Charged Oxime Reactivators on the HK-2 Cell Line in Renal Toxicity Screening
.
CHEMICAL RESEARCH IN TOXICOLOGY
. 34:699-703.
Full Text via DOI:
10.1021/acs.chemrestox.0c00489
Web of Science:
000630171600008
2021
Effects of novel 17β-hydroxysteroid dehydrogenase type 10 inhibitors on mitochondrial respiration
.
TOXICOLOGY LETTERS
. 339:12-19.
Full Text via DOI:
10.1016/j.toxlet.2020.12.012
Web of Science:
000608184700002
2021
Development of versatile and potent monoquaternary reactivators of acetylcholinesterase
.
ARCHIVES OF TOXICOLOGY
. 95:985-1001.
Full Text via DOI:
10.1007/s00204-021-02981-w
Web of Science:
000613184700001
2021
Molecular Modeling Studies on the Multistep Reactivation Process of Organophosphate-Inhibited Acetylcholinesterase and Butyrylcholinesterase
Full Text via DOI:
10.3390/biom11020169
Web of Science:
000622109100001
2021
Tacrine - Benzothiazoles: Novel class of potential multitarget anti-Alzheimets drugs dealing with cholinergic, amyloid and mitochondrial systems
.
BIOORGANIC CHEMISTRY
. 107.
Full Text via DOI:
10.1016/j.bioorg.2020.104596
Web of Science:
000618104800008
2021
Design, synthesis, and
in vitro
evaluation of BP-1-102 analogs with modified hydrophobic fragments for STAT3 inhibition
Full Text via DOI:
10.1080/14756366.2020.1871336
Web of Science:
000607423800001
2021
Pyridinium-2-carbaldoximes with quinolinium carboxamide moiety are simultaneous reactivators of acetylcholinesterase and butyrylcholinesterase inhibited by nerve agent surrogates
Full Text via DOI:
10.1080/14756366.2020.1869954
Web of Science:
000608910500001
2021
The Effect of Chemical Structure of OEG Ligand Shells with Quaternary Ammonium Moiety on the Colloidal Stabilization, Cellular Uptake and Photothermal Stability of Gold Nanorods
.
INTERNATIONAL JOURNAL OF NANOMEDICINE
. 16:3407-3427.
Full Text via DOI:
10.2147/IJN.S304953
Web of Science:
000651874100001
2020
Anticipated Social and Healthcare Economic Burden of People with Alzheimer's Disease in Two Selected Regions of the Czech Republic
Full Text via DOI:
10.3390/healthcare8040433
Web of Science:
000601427900001
2020
Glycosylated-imidazole aldoximes as reactivators of pesticides inhibited AChE: Synthesis and
in
-
vitro
reactivation study
.
ENVIRONMENTAL TOXICOLOGY AND PHARMACOLOGY
. 80.
Full Text via DOI:
10.1016/j.etap.2020.103454
Web of Science:
000583776900013
2020
Acetylcholinesterase Inhibition of Diversely Functionalized Quinolinones for Alzheimer's Disease Therapy
Full Text via DOI:
10.3390/ijms21113913
Web of Science:
000543400300175
2020
RNase T1 Refolding Assay for Determining Mitochondrial Cyclophilin D Activity: A Novel
In Vitro
Method Applicable in Drug Research and Discovery
.
BIOCHEMISTRY
. 59:1680-1687.
Full Text via DOI:
10.1021/acs.biochem.9b01025
Web of Science:
000530650400010
2020
A stereoselective approach in preparation of gamma-lactam precursors for oxazolomycin's synthesis
.
TETRAHEDRON
. 76.
Full Text via DOI:
10.1016/j.tet.2020.131111
Web of Science:
000525714700014
2020
Oxime K074-
in vitro
and
in silico
reactivation of acetylcholinesterase inhibited by nerve agents and pesticides
Full Text via DOI:
10.1080/15569543.2018.1485702
Web of Science:
000532601200007
2020
Benzothiazolyl Ureas are Low Micromolar and Uncompetitive Inhibitors of 17β-HSD10 with Implications to Alzheimer's Disease Treatment
Full Text via DOI:
10.3390/ijms21062059
Web of Science:
000529890200155
2020
Cysteine-Targeted Insecticides against
A
.
gambiae
Acetylcholinesterase Are Neither Selective nor Reversible Inhibitors
.
ACS MEDICINAL CHEMISTRY LETTERS
. 11:65-71.
Full Text via DOI:
10.1021/acsmedchemlett.9b00477
Web of Science:
000526400900010
2020
1,2,4-Triazole-based anticonvulsant agents with additional ROS scavenging activity are effective in a model of pharmacoresistant epilepsy
Full Text via DOI:
10.1080/14756366.2020.1748026
Web of Science:
000526646100001
2020
Synthesis,
in vitro
screening and molecular docking of isoquinolinium-5-carbaldoximes as acetylcholinesterase and butyrylcholinesterase reactivators
Full Text via DOI:
10.1080/14756366.2019.1710501
Web of Science:
000506063900001
2019
Highly hydrophilic cationic gold nanorods stabilized by novel quaternary ammonium surfactant with negligible cytotoxicity
.
JOURNAL OF BIOPHOTONICS
. 12.
Full Text via DOI:
10.1002/jbio.201900024
Web of Science:
000479453700001
2019
Pharmacokinetics of K117 and K127, two novel antidote candidates to treat Tabun poisoning
Full Text via DOI:
10.1016/j.cbi.2019.108737
Web of Science:
000482179600021
2019
Reactivation potency of two novel oximes (K456 and K733) against paraoxon-inhibited acetyl and butyrylcholinesterase:
In silico
and
in vitro
models
Full Text via DOI:
10.1016/j.cbi.2019.108735
Web of Science:
000482179600019
2019
Comparison of oximes K203 and K027 based on Benchmark dose analysis of rat diaphragmal acetylcholinesterase reactivation
Full Text via DOI:
10.1016/j.cbi.2019.05.034
Web of Science:
000474214200046
2019
Novel Benzothiazole-Based Ureas as 17β-HSD10 Inhibitors, A Potential Alzheimer's Disease Treatment
Full Text via DOI:
10.3390/molecules24152757
Web of Science:
000482441100080
2019
Surface screening, molecular modeling and
in vitro
studies on the interactions of aflatoxin M1 and human enzymes acetyl- and butyrylcholinesterase
Full Text via DOI:
10.1016/j.cbi.2019.05.022
Web of Science:
000474214200012
2019
Butyrylcholinesterase inhibited by nerve agents is efficiently reactivated with chlorinated pyridinium oximes
Full Text via DOI:
10.1016/j.cbi.2019.04.020
Web of Science:
000470976100003
2019
Experimental hydrophilic reactivator: bisoxime with three positive charges
Full Text via DOI:
10.1007/s11696-018-0612-6
Web of Science:
000459465100025
2019
Oxime K203: a drug candidate for the treatment of tabun intoxication
.
ARCHIVES OF TOXICOLOGY
. 93:673-691.
Full Text via DOI:
10.1007/s00204-018-2377-7
Web of Science:
000463730100009
2019
Comparison of Plasma and Brain Exposure Levels of Bis-pyridinium Oximes KR-22839 and KR-26256 with Asoxime and Obidoxime in Mice
Full Text via DOI:
10.1002/bkcs.11632
Web of Science:
000455598600001
2019
Donepezil plus chromone plus melatonin hybrids as promising agents for Alzheimer's disease therapy
Full Text via DOI:
10.1080/14756366.2018.1545766
Web of Science:
000457532600001
2019
Molecular modeling studies on the interactions of aflatoxin B1 and its metabolites with the peripheral anionic site of human acetylcholinesterase
.
JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS
. 37:2041-2048.
Full Text via DOI:
10.1080/07391102.2018.1475259
Web of Science:
000465025800010
2019
Synthesis and Biological Evaluation of Novel Chromone plus Donepezil Hybrids for Alzheimer's Disease Therapy
.
CURRENT ALZHEIMER RESEARCH
. 16:815-820.
Full Text via DOI:
10.2174/1567205016666191011112624
Web of Science:
000493721100004
2018
Pyridinium Oximes with
Ortho
-Positioned Chlorine Moiety Exhibit Improved Physicochemical Properties and Efficient Reactivation of Human Acetylcholinesterase Inhibited by Several Nerve Agents
.
JOURNAL OF MEDICINAL CHEMISTRY
. 61:10753-10766.
Full Text via DOI:
10.1021/acs.jmedchem.8b01398
Web of Science:
000453488200027
2018
Dose-response modeling of reactivating potency of oximes K027 and K203 against a direct acetylcholinesterase inhibitor in rat erythrocytes
.
FOOD AND CHEMICAL TOXICOLOGY
. 121:224-230.
Full Text via DOI:
10.1016/j.fct.2018.08.065
Web of Science:
000449242800023
2018
Molecular Modeling Studies on the Interactions of Aflatoxin B1 and Its Metabolites with Human Acetylcholinesterase. Part II: Interactions with the Catalytic Anionic Site (CAS)
Full Text via DOI:
10.3390/toxins10100389
Web of Science:
000448820400010
2018
Novel Group of AChE Reactivators-Synthesis, In Vitro Reactivation and Molecular Docking Study
Full Text via DOI:
10.3390/molecules23092291
Web of Science:
000447365100202
2018
QSAR Study of N-Myristoyltransferase Inhibitors of Antimalarial Agents
Full Text via DOI:
10.3390/molecules23092348
Web of Science:
000447365100259
2018
Synthesis, Biological Evaluation, and Docking Studies of Novel Bisquaternary Aldoxime Reactivators on Acetylcholinesterase and Butyrylcholinesterase Inhibited by Paraoxon
Full Text via DOI:
10.3390/molecules23051103
Web of Science:
000435204000118
2018
1-(Benzo[
d
]thiazol-2-yl)-3-phenylureas as dual inhibitors of casein kinase 1 and ABAD enzymes for treatment of neurodegenerative disorders
Full Text via DOI:
10.1080/14756366.2018.1445736
Web of Science:
000427559700001
2018
A newly developed oxime K203 is the most effective reactivator of tabun-inhibited acetylcholinesterase
Full Text via DOI:
10.1186/s40360-018-0196-3
Web of Science:
000425777700001
2018
Biological safety and tissue distribution of (16-mercaptohexadecyl) trimethylammonium bromide-modified cationic gold nanorods
.
BIOMATERIALS
. 154:275-290.
Full Text via DOI:
10.1016/j.biomaterials.2017.10.044
Web of Science:
000419538900022
2018
Effect of six oximes on acutely anticholinesterase inhibitor-induced oxidative stress in rat plasma and brain
.
ARCHIVES OF TOXICOLOGY
. 92:745-757.
Full Text via DOI:
10.1007/s00204-017-2101-z
Web of Science:
000425526000016
2018
Quantification through TLC-densitometric analysis, repellency and anticholinesterase activity of the homemade extract of Indian cloves
.
BIOMEDICAL CHROMATOGRAPHY
. 32.
Full Text via DOI:
10.1002/bmc.4096
Web of Science:
000423404000045
2018
In silico
and
in vitro
evaluation of two novel oximes (K378 and K727) in comparison to K-27 and pralidoxime against paraoxon-ethyl intoxication
.
TOXICOLOGY MECHANISMS AND METHODS
. 28:62-68.
Full Text via DOI:
10.1080/15376516.2017.1357777
Web of Science:
000418119300008
2018
In vitro
and
in silico
Evaluation of Non-Quaternary Reactivators of AChE as Antidotes of Organophosphorus Poisoning - a New Hope or a Blind Alley?
Full Text via DOI:
10.2174/1573406414666180112105657
Web of Science:
000429554400008
2018
Development of small bisquaternary cholinesterase inhibitors as drugs for pre-treatment of nerve agent poisonings
Full Text via DOI:
10.2147/DDDT.S133038
Web of Science:
000427385300001
2018
Oxime K033-reactivation Activity of Cholinesterases Inhibited by Various Nerve Agents and Organophosphorus Pesticides
Full Text via DOI:
10.2174/1570164615666180713112238
Web of Science:
000445684700001
2017
Pharmacokinetic profile of promising acetylcholinesterase reactivators K027 and K203 in experimental pigs
.
TOXICOLOGY LETTERS
. 273:20-25.
Full Text via DOI:
10.1016/j.toxlet.2017.03.017
Web of Science:
000400459600003
2017
Synthesis and evaluation of frentizole-based indolyl thiourea analogues as MAO/ABAD inhibitors for Alzheimer's disease treatment
.
BIOORGANIC & MEDICINAL CHEMISTRY
. 25:1143-1152.
Full Text via DOI:
10.1016/j.bmc.2016.12.029
Web of Science:
000394201900031
2017
6-Benzothiazolyl Ureas, Thioureas and Guanidines are Potent Inhibitors of ABAD/17
β
-HSD10 and Potential Drugs for Alzheimer's Disease Treatment: Design, Synthesis and
in vitro
Evaluation
Full Text via DOI:
10.2174/1573406413666170109142725
Web of Science:
000402479000004
2017
A comparison of the reactivating and therapeutic efficacy of two novel bispyridinium oximes (K305, K307) with the oxime K203 and trimedoxime in tabun-poisoned rats and mice
.
JOURNAL OF APPLIED BIOMEDICINE
. 15:49-53.
Full Text via DOI:
10.1016/j.jab.2016.09.008
Web of Science:
000396404200007
2017
Alzheimer's Disease Drugs- In Vitro Comparison of Cholinesterase Inhibition and beta-amyloid Modulation
Full Text via DOI:
10.2174/1570180814666161228143846
Web of Science:
000404984700013
2017
Bis-isoquinolinium and bis-pyridinium acetylcholinesterase inhibitors: in vitro screening of probes for novel selective insecticides
.
RSC ADVANCES
. 7:39279-39291.
Full Text via DOI:
10.1039/c7ra05838a
Web of Science:
000407762300063
2017
Progress in acetylcholinesterase reactivators and in the treatment of organophosphorus intoxication: a patent review (2006-2016)
Full Text via DOI:
10.1080/13543776.2017.1338275
Web of Science:
000407436800001
2017
Tetroxime: reactivation potency - in vitro and in silico study
.
RSC ADVANCES
. 7:7041-7045.
Full Text via DOI:
10.1039/c6ra16499d
Web of Science:
000393756000030
2016
Two-Step Mechanism of Cellular Uptake of Cationic Gold Nanoparticles Modified by (16-Mercaptohexadecyl)trimethylammonium Bromide
.
BIOCONJUGATE CHEMISTRY
. 27:2558-2574.
Full Text via DOI:
10.1021/acs.bioconjchem.6b00491
Web of Science:
000385992000039
2016
Design, synthesis and in vitro evaluation of benzothiazole-based ureas as potential ABAD/17β-HSD10 modulators for Alzheimer's disease treatment
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
. 26:3675-3678.
Full Text via DOI:
10.1016/j.bmcl.2016.05.087
Web of Science:
000380574100058
2016
Therapeutic and reactivating efficacy of oximes K027 and K203 against a direct acetylcholinesterase inhibitor
.
NEUROTOXICOLOGY
. 55:33-39.
Full Text via DOI:
10.1016/j.neuro.2016.05.006
Web of Science:
000380385800005
2016
Design, Synthesis and in vitro Evaluation of Indolotacrine Analogues as Multitarget-Directed Ligands for the Treatment of Alzheimer's Disease
.
CHEMMEDCHEM
. 11:1264-1269.
Full Text via DOI:
10.1002/cmdc.201500383
Web of Science:
000380024300010
2016
Oxime-mediated in vitro reactivation kinetic analysis of organophosphates-inhibited human and electric eel acetylcholinesterase
.
TOXICOLOGY MECHANISMS AND METHODS
. 26:319-326.
Full Text via DOI:
10.3109/15376516.2016.1143070
Web of Science:
000380053100002
2016
Investigation of the reactivation kinetics of a large series of bispyridinium oximes with organophosphate-inhibited human acetylcholinesterase
.
TOXICOLOGY LETTERS
. 244:136-142.
Full Text via DOI:
10.1016/j.toxlet.2015.07.007
Web of Science:
000369704400019
2016
Small Quaternary Inhibitors K298 and K524: Cholinesterases Inhibition, Absorption, Brain Distribution, and Toxicity
Full Text via DOI:
10.1007/s12640-015-9582-4
Web of Science:
000368194200008
2016
Development and validation of a FIA/UV-vis method for p
K
a
determination of oxime based acetylcholinesterase reactivators
Full Text via DOI:
10.1016/j.jpba.2015.09.010
Web of Science:
000365145500030
2016
A 7-methoxytacrine-4-pyridinealdoxime hybrid as a novel prophylactic agent with reactivation properties in organophosphate intoxication
.
TOXICOLOGY RESEARCH
. 5:1012-1016.
Full Text via DOI:
10.1039/c6tx00130k
Web of Science:
000378716100003
2016
Monooxime Bispyridinium Reactivators Bearing Xylene Linker Synthesis and In Vitro Evaluation on Model of Organophosphate-Inhibited Acetylcholinesterase
Full Text via DOI:
10.2174/1573406411666151002125640
Web of Science:
000376450400006
2016
TRISOXIME - a Bulky Trisquaternary Reactivator of Acetylcholinesterase
Full Text via DOI:
10.2174/1570180812666150923235240
Web of Science:
000374883700003
2015
A comparison of the reactivating and therapeutic efficacy of two novel bispyridinium oximes (K920, K923) with the oxime K203 and trimedoxime in tabun-poisoned rats and mice
.
JOURNAL OF APPLIED BIOMEDICINE
. 13:299-304.
Full Text via DOI:
10.1016/j.jab.2015.07.002
Web of Science:
000362983300006
2015
Flavones Inhibit the Activity of AKR1B10, a Promising Therapeutic Target for Cancer Treatment
.
JOURNAL OF NATURAL PRODUCTS
. 78:2666-2674.
Full Text via DOI:
10.1021/acs.jnatprod.5b00616
Web of Science:
000366005800020
2015
Comparative determination of the efficacy of bispyridinium oximes in paraoxon poisoning
.
ARHIV ZA HIGIJENU RADA I TOKSIKOLOGIJU-ARCHIVES OF INDUSTRIAL HYGIENE AND TOXICOLOGY
. 66:129-134.
Full Text via DOI:
10.1515/aiht-2015-66-2623
Web of Science:
000358360900004
2015
Design, synthesis and in vitro testing of 7-methoxytacrine-amantadine analogues: a novel cholinesterase inhibitors for the treatment of Alzheimer's disease
Full Text via DOI:
10.1007/s00044-015-1316-x
Web of Science:
000355933000031
2015
Preparation of 7-Methoxy Tacrine Dimer Analogs and Their In vitro/In silico Evaluation as Potential Cholinesterase Inhibitors
Full Text via DOI:
10.1002/bkcs.10317
Web of Science:
000355986100017
2015
Catalytic Soman Scavenging by the Y337A/F338A Acetylcholinesterase Mutant Assisted with Novel Site-Directed Aldoximes
.
CHEMICAL RESEARCH IN TOXICOLOGY
. 28:1036-1044.
Full Text via DOI:
10.1021/acs.chemrestox.5b00060
Web of Science:
000354907500021
2015
A Comparison of the Reactivating and Therapeutic Efficacy of Two Newly Developed Oximes (K727 and K733) with Oxime K203 and Trimedoxime in Tabun-Poisoned Rats and Mice
Full Text via DOI:
10.1111/bcpt.12327
Web of Science:
000351367600012
2015
A comparison of the reactivating and therapeutic efficacy of two novel bispyridinium oximes (K727, K733) with the oxime HI-6 and obidoxime in sarin-poisoned rats and mice
.
TOXICOLOGY MECHANISMS AND METHODS
. 25:229-233.
Full Text via DOI:
10.3109/15376516.2015.1036333
Web of Science:
000355988300009
2015
Ligand-based 3D QSAR analysis of reactivation potency of mono- and bis-pyridinium aldoximes toward VX-inhibited rat acetylcholinesterase
Full Text via DOI:
10.1016/j.jmgm.2014.11.010
Web of Science:
000350088600012
2015
Reactivation kinetics of 31 structurally different bispyridinium oximes with organophosphate-inhibited human butyrylcholinesterase
.
ARCHIVES OF TOXICOLOGY
. 89:405-414.
Full Text via DOI:
10.1007/s00204-014-1288-5
Web of Science:
000350030200009
2015
A Direct Interaction Between Mitochondrial Proteins and Amyloid-β Peptide and its Significance for the Progression and Treatment of Alzheimer's Disease
.
CURRENT MEDICINAL CHEMISTRY
. 22:1056-1085.
Full Text via DOI:
10.2174/0929867322666150114163051
Web of Science:
000350477600002
2015
Benzothiazoles - Scaffold of Interest for CNS Targeted Drugs
.
CURRENT MEDICINAL CHEMISTRY
. 22:730-747.
Full Text via DOI:
10.2174/0929867322666141212120631
Web of Science:
000349388600006
2015
Kinetic and physicochemical analysis of structurally different bis-pyridinium oximes against pesticide inhibited AChE
Web of Science:
000348245200005
2015
Preparation,
In Vitro
Screening and Molecular Modelling of Monoquaternary Compounds Related to the Selective Acetylcholinesterase Inhibitor BW284c51
Web of Science:
000349330100004
2015
Universality of Oxime K203 for Reactivation of Nerve Agent-Inhibited AChE
Full Text via DOI:
10.2174/1573406411666150407154204
Web of Science:
000361825400011
2014
6-Hydroxyquinolinium salts differing in the length of alkyl side-chain: Synthesis and antimicrobial activity
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
. 24:5238-5241.
Full Text via DOI:
10.1016/j.bmcl.2014.09.060
Web of Science:
000343901400021
2014
Structural modifications of dicationic acetylcholinesterase reactivators studied under ion-pairing mechanism in reversed-phase liquid chromatography
.
JOURNAL OF SEPARATION SCIENCE
. 37:3024-3032.
Full Text via DOI:
10.1002/jssc.201400390
Web of Science:
000344250300002
2014
Assessment of antidotal efficacy of cholinesterase reactivators against paraoxon: In vitro reactivation kinetics and physicochemical properties
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
. 24:4743-4748.
Full Text via DOI:
10.1016/j.bmcl.2014.07.095
Web of Science:
000342574600024
2014
7-MEOTA-donepezil like compounds as cholinesterase inhibitors: Synthesis, pharmacological evaluation, molecular modeling and QSAR studies
.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
. 82:426-438.
Full Text via DOI:
10.1016/j.ejmech.2014.05.066
Web of Science:
000339039100040
2014
Cholinergic antagonist 3-quinuclidinyl benzilate - Impact on learning and memory in Wistar rats
.
BEHAVIOURAL BRAIN RESEARCH
. 266:193-200.
Full Text via DOI:
10.1016/j.bbr.2014.03.001
Web of Science:
000335805300025
2014
In Vivo
Evaluation of Cholinesterase Activity, Oxidative Stress Markers, Cyto- and Genotoxicity of K048 Oxime - a Promising Antidote against Organophosphate Poisoning
Full Text via DOI:
10.1111/bcpt.12158
Web of Science:
000332208300008
2014
Interaction of cholinesterase modulators with DNA and their cytotoxic activity
.
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES
. 64:53-62.
Full Text via DOI:
10.1016/j.ijbiomac.2013.11.022
Web of Science:
000334147300009
2014
Retention Behavior of Pyridinium Oximes on PFP Stationary Phase in High-Performance Liquid Chromatography
Full Text via DOI:
10.1093/chromsci/bmt019
Web of Science:
000342734000009
2014
The evaluation of the reactivating and therapeutic efficacy of two novel oximes (K361 and K378) in comparison with the oxime K203 and trimedoxime in tabun-poisoned rats and mice
.
TOXICOLOGY MECHANISMS AND METHODS
. 24:173-178.
Full Text via DOI:
10.3109/15376516.2013.871766
Web of Science:
000332116900002
2014
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