European Journal of Medicinal Chemistry

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European Journal of Medicinal Chemistry Journal

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Novel D2/5-HT receptor modulators related to cariprazine with potential implication to schizophrenia treatment. 232. 2022
Design of gp120 HIV-1 entry inhibitors by scaffold hopping via isosteric replacements. 224. 2021
Diaryl hydroxylamines as pan or dual inhibitors of indoleamine 2,3-dioxygenase-1, indoleamine 2,3-dioxygenase-2 and tryptophan dioxygenase. 162:455-464. 2019
Optimization of the first small-molecule relaxin/insulin-like family peptide receptor (RXFP1) agonists: Activation results in an antifibrotic gene expression profile. 156:79-92. 2018
Structure-based lead optimization to improve antiviral potency and ADMET properties of phenyl-1H-pyrrole-carboxamide entry inhibitors targeted to HIV-1 gp120. 154:367-391. 2018
The 4-N-acyl and 4-N-alkyl gemcitabine analogues with silicon-fluoride-acceptor: Application to ¹⁸F-Radiolabeling. 148:314-324. 2018
Synthesis, evaluation, and CoMFA study of fluoroquinophenoxazine derivatives as bacterial topoisomerase IA inhibitors. 125:515-527. 2017
Design and synthesis of bis(indolyl)ketohydrazide-hydrazones: Identification of potent and selective novel tubulin inhibitors. 136:184-194. 2017
Bicyclic octahydrocyclohepta[b]pyrrol-4(1H)one derivatives as novel selective anti-hepatitis C virus agents. 122:319-325. 2016
Discovery of the 2-phenyl-4,5,6,7-Tetrahydro-1H-indole as a novel anti-hepatitis C virus targeting scaffold. 96:250-258. 2015
Synthesis and biological evaluations of novel endomorphin analogues containing α-hydroxy-β-phenylalanine (AHPBA) displaying mixed μ/δ opioid receptor agonist and δ opioid receptor antagonist activities. 92:270-281. 2015
7-MEOTA-donepezil like compounds as cholinesterase inhibitors: Synthesis, pharmacological evaluation, molecular modeling and QSAR studies. 82:426-438. 2014
Ligand/kappa-opioid receptor interactions: Insights from the X-ray crystal structure. 66:114-121. 2013
Synthesis and biological evaluation of 2-indolinone derivatives as potential antitumor agents. 46:5970-5977. 2011
Preparation and in vitro screening of symmetrical bis-isoquinolinium cholinesterase inhibitors bearing various connecting linkage - Implications for early Myasthenia gravis treatment. 46:811-818. 2011
Synthesis of functionalized tetrasubstituted pyrazolyl heterocycles - A review 2011
Recent methodologies toward the synthesis of valdecoxib: A potential 3,4-diarylisoxazolyl COX-II inhibitor 2010
2,6-Bis-arylmethyloxy-5-hydroxychromones with antiviral activity against both hepatitis C virus (HCV) and SARS-associated coronavirus (SCV). 2011

International Standard Serial Number (ISSN)

0223-5234

Electronic International Standard Serial Number (EISSN)

1768-3254