Design of gp120 HIV-1 entry inhibitors by scaffold hopping via isosteric replacements Article

Iusupov, Ildar R, Curreli, Francesca, Spiridonov, Evgeniy A et al. (2021). Design of gp120 HIV-1 entry inhibitors by scaffold hopping via isosteric replacements . EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 224 10.1016/j.ejmech.2021.113681

Open Access International Collaboration

cited authors

  • Iusupov, Ildar R; Curreli, Francesca; Spiridonov, Evgeniy A; Markov, Pavel O; Ahmed, Shahad; Belov, Dmitry S; Manasova, Ekaterina; Altieri, Andrea; Kurkin, Alexander; Debnath, Asim K

sustainable development goals

authors

publication date

  • July 8, 2021

keywords

  • ACCURATE DOCKING
  • ANTIVIRAL ACTIVITY
  • BINDING
  • Chemistry, Medicinal
  • DISCOVERY
  • DIVERSITY
  • Drug discovery
  • GLIDE
  • HIV
  • Lead optimization
  • Life Sciences & Biomedicine
  • OPTIMIZATION
  • Pharmacology & Pharmacy
  • RATIONAL DESIGN
  • SMALL-MOLECULE HIV-1
  • Science & Technology
  • Screening
  • Synthesis
  • TARGET
  • gp120

Digital Object Identifier (DOI)

publisher

  • ELSEVIER FRANCE-EDITIONS SCIENTIFIQUES MEDICALES ELSEVIER

volume

  • 224