Florida International University
Edit Your Profile
FIU Discovery
Toggle navigation
Browse
Home
People
Organizations
Scholarly & Creative Works
Research Facilities
Support
Edit Your Profile
Belov, Dmitrii
Share this page
Twitter
Email
Copy link
Share
Scholarly & Creative Works
Identifiers
View All
Scholarly & Creative Works
selected scholarly works & creative activities
Article
2021
Design of gp120 HIV-1 entry inhibitors by scaffold hopping via isosteric replacements
.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
. 224.
Full Text via DOI:
10.1016/j.ejmech.2021.113681
Web of Science:
000703110000010
2021
Synthesis of Vanadium Oxo Alkylidene Complex and Its Reactivity in Ring-Closing Olefin Metathesis Reactions
.
ORGANOMETALLICS
. 40:2939-2944.
Full Text via DOI:
10.1021/acs.organomet.1c00425
Web of Science:
000696376900004
2021
Ring-Closing Olefin Metathesis Catalyzed by Well-Defined Vanadium Alkylidene Complexes
.
CHEMISTRY-A EUROPEAN JOURNAL
. 27:4578-4582.
Full Text via DOI:
10.1002/chem.202005438
Web of Science:
000614766300001
2021
Design, synthesis, and antiviral activity of a series of CD4-mimetic small-molecule HIV-1 entry inhibitors
.
BIOORGANIC & MEDICINAL CHEMISTRY
. 32.
Full Text via DOI:
10.1016/j.bmc.2021.116000
Web of Science:
000616056900008
2021
Stereospecific Ring-Opening Metathesis Polymerization of Norbornene Catalyzed by Iron Complexes
.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
. 60:2934-2938.
Full Text via DOI:
10.1002/anie.202011150
Web of Science:
000597161900001
2021
Stereospecific Ring‐Opening Metathesis Polymerization of Norbornene Catalyzed by Iron Complexes
Full Text via DOI:
10.1002/ange.202011150
2020
Preclinical Optimization of gp120 Entry Antagonists as anti-HIV-1 Agents with Improved Cytotoxicity and ADME Properties through Rational Design, Synthesis, and Antiviral Evaluation
.
JOURNAL OF MEDICINAL CHEMISTRY
. 63:1724-1749.
Full Text via DOI:
10.1021/acs.jmedchem.9b02149
Web of Science:
000517673100020
2018
Synthesis, Antiviral Activity, and Structure-Activity Relationship of 1,3-Benzodioxolyl Pyrrole-Based Entry Inhibitors Targeting the Phe43 Cavity in HIV-1 gp120
.
CHEMMEDCHEM
. 13:2332-2348.
Full Text via DOI:
10.1002/cmdc.201800534
Web of Science:
000449679800009
2018
Structure-based lead optimization to improve antiviral potency and ADMET properties of phenyl-1H-pyrrole-carboxamide entry inhibitors targeted to HIV-1 gp120
.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
. 154:367-391.
Full Text via DOI:
10.1016/j.ejmech.2018.04.062
Web of Science:
000437551600029
2018
Guanidine-Containing Phenyl-Pyrrole Compounds as Probes for Generating HIV Entry Inhibitors Targeted to gp120
.
CHEMISTRYSELECT
. 3:6450-6453.
Full Text via DOI:
10.1002/slct.201801662
Web of Science:
000435933100025
2017
A Small-Molecule Inhibitor of Prion Replication and Mutant Prion Protein Toxicity
.
CHEMMEDCHEM
. 12:1286-1292.
Full Text via DOI:
10.1002/cmdc.201700302
Web of Science:
000429592300007
2017
Synthesis of 5-Arylpyrrole-2-carboxylic Acids as Key Intermediates for NBD Series HIV-1 Entry Inhibitors
.
SYNTHESIS-STUTTGART
. 49:3692-3699.
Full Text via DOI:
10.1055/s-0036-1588780
Web of Science:
000407139300019
2017
Synthesis, Antiviral Potency, in Vitro ADMET, and X-ray Structure of Potent CD4 Mimics as Entry Inhibitors That Target the Phe43 Cavity of HIV-1 gp120
.
JOURNAL OF MEDICINAL CHEMISTRY
. 60:3124-3153.
Full Text via DOI:
10.1021/acs.jmedchem.7b00179
Web of Science:
000399436100035
2016
Design, synthesis and evaluation of small molecule CD4-mimics as entry inhibitors possessing broad spectrum anti-HIV-1 activity
.
BIOORGANIC & MEDICINAL CHEMISTRY
. 24:5988-6003.
Full Text via DOI:
10.1016/j.bmc.2016.09.057
Web of Science:
000387200000031
2016
Bicyclic octahydrocyclohepta[b]pyrrol-4(1H)one derivatives as novel selective anti-hepatitis C virus agents
.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
. 122:319-325.
Full Text via DOI:
10.1016/j.ejmech.2016.06.041
Web of Science:
000383003900027
2016
Fragment-Based Discovery of 5-Arylisatin-Based Inhibitors of Matrix Metalloproteinases 2 and 13
.
CHEMMEDCHEM
. 11:1892-1898.
Full Text via DOI:
10.1002/cmdc.201600266
Web of Science:
000383610100003
2016
ChemInform Abstract: Oxidative Dearomatization of 4,5,6,7‐Tetrahydro‐1H‐indoles Obtained by Metal‐ and Solvent‐Free Thermal 5‐endo‐dig Cyclization: The Route to Erythrina and Lycorine Alkaloids.
Full Text via DOI:
10.1002/chin.201641135
2016
Oxidative Dearomatization of 4,5,6,7-Tetrahydro-1
H
-indoles Obtained by Metal- and Solvent-Free Thermal 5-
endo
-
dig
Cyclization: The Route to Erythrina and Lycorine Alkaloids
.
CHEMISTRY-A EUROPEAN JOURNAL
. 22:7262-7267.
Full Text via DOI:
10.1002/chem.201600273
Web of Science:
000377604100038
2015
Structure-Based Design of a Small Molecule CD4-Antagonist with Broad Spectrum Anti-HIV-1 Activity
.
JOURNAL OF MEDICINAL CHEMISTRY
. 58:6909-6927.
Full Text via DOI:
10.1021/acs.jmedchem.5b00709
Web of Science:
000361254600013
2015
ChemInform Abstract: Synthesis of Bicyclic Proline Derivatives by the Aza‐Cope—Mannich Reaction: Formal Synthesis of (.+‐.)‐Acetylaranotin.
Full Text via DOI:
10.1002/chin.201528255
2015
Discovery of the 2-phenyl-4,5,6,7-Tetrahydro-1
H
-indole as a novel anti-hepatitis C virus targeting scaffold
.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
. 96:250-258.
Full Text via DOI:
10.1016/j.ejmech.2015.04.022
Web of Science:
000355712500024
2015
Synthesis of Bicyclic Proline Derivatives by the Aza-Cope-Mannich Reaction: Formal Synthesis of (±)-Acetylaranotin
.
CHEMISTRY-A EUROPEAN JOURNAL
. 21:4141-4147.
Full Text via DOI:
10.1002/chem.201405811
Web of Science:
000350762400037
2014
ChemInform Abstract: An Effective Activation of Palladium Phosphine Complexes in Aqueous Phase Reactions of Hetero‐Aromatic Boronic Acids with Aryl Halides.
Full Text via DOI:
10.1002/chin.201439057
2014
ChemInform Abstract: Synthesis of Non‐Natural L‐Alanine Derivatives Using the Aza‐Cope—Mannich Reaction.
Full Text via DOI:
10.1002/chin.201437211
2014
An Effective Activation of Palladium Phosphine Complexes in Aqueous Phase Reactions of Hetero-Aromatic Boronic Acids with Aryl Halides
Full Text via DOI:
10.1007/s10593-014-1443-1
Web of Science:
000334271700004
2014
Synthesis of non-natural L-alanine derivatives using the aza-Cope-Mannich reaction
.
TETRAHEDRON-ASYMMETRY
. 25:468-472.
Full Text via DOI:
10.1016/j.tetasy.2014.01.011
Web of Science:
000334985000011
2013
ChemInform Abstract: Synthesis of 4,5,6,7‐Tetrahydro‐1H‐indole Derivatives Through Successive Sonogashira Coupling/Pd‐Mediated 5‐endo‐dig Cyclization.
Full Text via DOI:
10.1002/chin.201324090
2013
ChemInform Abstract: Highly Stereoselective and Scalable Synthesis of trans‐Fused Octahydrocyclohepta[b]pyrrol‐4(1H)‐ones via the Aza‐Cope—Mannich Rearrangement in Racemic and Enantiopure Forms.
Full Text via DOI:
10.1002/chin.201316078
2013
Synthesis of 4,5,6,7-Tetrahydro-1H-indole Derivatives Through Successive Sonogashira Coupling/Pd-Mediated 5-endo-dig Cyclization
.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
. 2013:649-652.
Full Text via DOI:
10.1002/ejoc.201201417
Web of Science:
000316193000002
2012
Highly Stereoselective and Scalable Synthesis of trans-Fused Octahydrocyclohepta[b]pyrrol-4(1H)-ones via the Aza-Cope-Mannich Rearrangement in Racemic and Enantiopure Forms
.
JOURNAL OF ORGANIC CHEMISTRY
. 77:10125-10134.
Full Text via DOI:
10.1021/jo301762a
Web of Science:
000311073000020
2012
ChemInform Abstract: Palladium‐Catalyzed Carboamination in the Synthesis of Nitrogen‐Containing Heterocycles
Full Text via DOI:
10.1002/chin.201233248
2012
(1
R
, 3
R
,3aS,8a
R
)-4-Oxo-3-phenyl-1-[(1
R
)1-phenylethyl] decahydrocyclohepta[
b
]pyrrol-1-ium bromide
Full Text via DOI:
10.1107/S1600536812028073
Web of Science:
000421522300358
2012
Palladium-catalyzed carboamination in the synthesis of nitrogen-containing heterocycles
Full Text via DOI:
10.1007/s10593-012-0971-9
Web of Science:
000304163900014
2011
Synthesis of (3RS,3aSR,8aSR)-3-phenyloctahydrocyclohepta[b]pyrrol-4(1H)-one via the aza-Cope-Mannich rearrangement
.
TETRAHEDRON
. 67:9214-9218.
Full Text via DOI:
10.1016/j.tet.2011.09.047
Web of Science:
000296988800023
2009
ChemInform Abstract: tert‐Butyl (2S)‐(p‐Tolylsulfonyloxy)propionate (II) — A Suitable Reagent for the Direct Alkylation of Indole Derivatives.
Full Text via DOI:
10.1002/chin.200924112
2008
Tert-Butyl (25)-(4-methylphenylsulfonyloxy)propionate - Convenient reagent for the direct alkylation of indole derivatives
2008
tert-Butyl (2S)-(p-tolylsulfonyloxy)propionate - a suitable reagent for the direct alkylation of indole derivatives
Full Text via DOI:
10.1007/s10593-008-0160-z
Web of Science:
000261622600010
Other Scholarly Work
2017
Correction to Synthesis, Antiviral Potency, in Vitro ADMET, and X-ray Structure of Potent CD4 Mimics as Entry Inhibitors That Target the Phe43 Cavity of HIV-1 gp120.
.
JOURNAL OF MEDICINAL CHEMISTRY
. 4734.
Full Text via DOI:
10.1021/acs.jmedchem.7b00690
2015
Synthesis of bicyclic proline derivatives by the aza-Cope-Mannich reaction: formal synthesis of (±)-acetylaranotin.
.
CHEMISTRY-A EUROPEAN JOURNAL
. 4141-4147.
Full Text via DOI:
10.1002/chem.201405811
Review
2021
Olefin Metathesis by First-Row Transition Metals
. 924-937.
Full Text via DOI:
10.1002/cplu.202100192
Web of Science:
000674289400022
Identifiers
ORCID iD
https://orcid.org/0000-0002-1338-4184
(confirmed)
visualizations
Co-author Network
Map of Science