Synthesis, Antiviral Potency, in Vitro ADMET, and X-ray Structure of Potent CD4 Mimics as Entry Inhibitors That Target the Phe43 Cavity of HIV-1 gp120 Article

Curreli, Francesca, Kwon, Young Do, Belov, Dmitry S et al. (2017). Synthesis, Antiviral Potency, in Vitro ADMET, and X-ray Structure of Potent CD4 Mimics as Entry Inhibitors That Target the Phe43 Cavity of HIV-1 gp120 . JOURNAL OF MEDICINAL CHEMISTRY, 60(7), 3124-3153. 10.1021/acs.jmedchem.7b00179

International Collaboration

cited authors

  • Curreli, Francesca; Kwon, Young Do; Belov, Dmitry S; Ramesh, Ranjith R; Kurkin, Alexander V; Altieri, Andrea; Kwong, Peter D; Debnath, Asim K

sustainable development goals

authors

publication date

  • April 13, 2017

published in

keywords

  • BINDING
  • CCR5 CORECEPTOR
  • Chemistry, Medicinal
  • EARLY SUBTYPE
  • ENV CLONES
  • ENVELOPE
  • IMMUNODEFICIENCY-VIRUS TYPE-1
  • Life Sciences & Biomedicine
  • METABOLISM
  • NEUTRALIZATION
  • Pharmacology & Pharmacy
  • SMALL-MOLECULE INHIBITORS
  • STRUCTURE-BASED DESIGN
  • Science & Technology

Digital Object Identifier (DOI)

publisher

  • AMER CHEMICAL SOC

start page

  • 3124

end page

  • 3153

volume

  • 60

issue

  • 7