Bioorganic and Medicinal Chemistry

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Bioorganic and Medicinal Chemistry Journal

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Design, synthesis, and antiviral activity of a series of CD4-mimetic small-molecule HIV-1 entry inhibitors. 32. 2021
4-N-Alkanoyl and 4-N-alkyl gemcitabine analogues with NOTA chelators for 68-gallium labelling. 26:5624-5630. 2018
Synthesis and evaluation of frentizole-based indolyl thiourea analogues as MAO/ABAD inhibitors for Alzheimer's disease treatment. 25:1143-1152. 2017
Synthesis, evaluation and molecular modelling studies of 2-(carbazol-3-yl)-2-oxoacetamide analogues as a new class of potential pancreatic lipase inhibitors. 25:609-620. 2017
Design, synthesis and evaluation of small molecule CD4-mimics as entry inhibitors possessing broad spectrum anti-HIV-1 activity. 24:5988-6003. 2016
Exploration of bivalent ligands targeting putative mu opioid receptor and chemokine receptor CCR5 dimerization. 24:5969-5987. 2016
Identification of 5,6-dihydroimidazo[2,1-b]thiazoles as a new class of antimicrobial agents. 24:5633-5638. 2016
The structures of three metabolites of the algal hepatotoxin okadaic acid produced by oxidation with human cytochrome P450. 20:3742-3745. 2012
A bright approach to the immunoproteasome: Development of LMP2/β1i-specific imaging probes. 20:607-613. 2012
Oxidative folding of lysozyme with aromatic dithiols, and aliphatic and aromatic monothiols. 20:1020-1028. 2012
Inhibition of LuxS by S-ribosylhomocysteine analogues containing a [4-aza]ribose ring. 19:5507-5519. 2011
Substituted lactam and cyclic azahemiacetals modulate Pseudomonas aeruginosa quorum sensing. 19:5500-5506. 2011
Mono-oxime bisquaternary acetylcholinesterase reactivators with prop-1,3-diyl linkage-Preparation, in vitro screening and molecular docking. 19:754-762. 2011
Towards a systematic characterization of the antiprotozoal activity landscape of benzimidazole derivatives. 18:7380-7391. 2010
Inhibition of S-ribosylhomocysteinase (LuxS) by substrate analogues modified at the ribosyl C-3 position. 17:6699-6706. 2009
Fluorinated pyridinium oximes as potential reactivators for acetylcholinesterases inhibited by paraoxon organophosphorus agent. 17:6213-6217. 2009
Identification, structure-activity relationships and molecular modeling of potent triamine and piperazine opioid ligands. 17:5583-5597. 2009
Monoquaternary pyridinium salts with modified side chain - synthesis and evaluation on model of tabun- and paraoxon-inhibited acetylcholinesterase. 16:8218-8223. 2008
Conformation-opioid activity relationships of bicyclic guanidines from 3D similarity analysis. 16:5932-5938. 2008
Synthesis of 5′-functionalized nucleosides:: S-Adenosylhomocysteine analogues with the carbon-5′ and sulfur atoms replaced by a vinyl or halovinyl unit. 16:5424-5433. 2008
S-ribosylhomocysteine analogues with the carbon-5 and sulfur atoms replaced by a vinyl or (fluoro)vinyl unit. 16:5090-5102. 2008
Rate enhancement of the oxidative folding of lysozyme by the use of aromatic thiol containing redox buffers. 16:2579-2590. 2008
Monooxime reactivators of acetylcholinesterase with (E)-but-2-ene linker -: Preparation and reactivation of tabun- and paraoxon-inhibited acetylcholinesterase. 15:6733-6741. 2007
Lead optimization of 7-benzyloxy 2-(4′-pyridylmethyl)thio isoflavone aromatase inhibitors. 13:6571-6577. 2005
Synthesis and characterization of azole isoflavone inhibitors of aromatase. 13:4063-4070. 2005
Identification of novel small-molecule Ulex europaeus I mimetics for targeted drug delivery. 11:4991-4997. 2003
The structural basis for kainoid selectivity at AMPA receptors revealed by low-mode docking calculations. 11:551-559. 2003
The synthesis of peptidomimetic combinatorial libraries through successive amide alkylations 1996

International Standard Serial Number (ISSN)

0968-0896

Electronic International Standard Serial Number (EISSN)

1464-3391