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BIOORGANIC & MEDICINAL CHEMISTRY
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Overview
publication venue for
Design, synthesis, and antiviral activity of a series of CD4-mimetic small-molecule HIV-1 entry inhibitors
. 32.
2021
4-N-Alkanoyl and 4-N-alkyl gemcitabine analogues with NOTA chelators for 68-gallium labelling
. 26:5624-5630.
2018
Synthesis and evaluation of frentizole-based indolyl thiourea analogues as MAO/ABAD inhibitors for Alzheimer's disease treatment
. 25:1143-1152.
2017
Synthesis, evaluation and molecular modelling studies of 2-(carbazol-3-yl)-2-oxoacetamide analogues as a new class of potential pancreatic lipase inhibitors
. 25:609-620.
2017
Design, synthesis and evaluation of small molecule CD4-mimics as entry inhibitors possessing broad spectrum anti-HIV-1 activity
. 24:5988-6003.
2016
Exploration of bivalent ligands targeting putative mu opioid receptor and chemokine receptor CCR5 dimerization
. 24:5969-5987.
2016
Identification of 5,6-dihydroimidazo[2,1-b]thiazoles as a new class of antimicrobial agents
. 24:5633-5638.
2016
The structures of three metabolites of the algal hepatotoxin okadaic acid produced by oxidation with human cytochrome P450
. 20:3742-3745.
2012
A bright approach to the immunoproteasome: Development of LMP2/β1i-specific imaging probes
. 20:607-613.
2012
Oxidative folding of lysozyme with aromatic dithiols, and aliphatic and aromatic monothiols
. 20:1020-1028.
2012
Inhibition of LuxS by
S
-ribosylhomocysteine analogues containing a [4-aza]ribose ring
. 19:5507-5519.
2011
Substituted lactam and cyclic azahemiacetals modulate
Pseudomonas aeruginosa
quorum sensing
. 19:5500-5506.
2011
Mono-oxime bisquaternary acetylcholinesterase reactivators with prop-1,3-diyl linkage-Preparation, in vitro screening and molecular docking
. 19:754-762.
2011
Towards a systematic characterization of the antiprotozoal activity landscape of benzimidazole derivatives
. 18:7380-7391.
2010
Inhibition of S-ribosylhomocysteinase (LuxS) by substrate analogues modified at the ribosyl C-3 position
. 17:6699-6706.
2009
Fluorinated pyridinium oximes as potential reactivators for acetylcholinesterases inhibited by paraoxon organophosphorus agent
. 17:6213-6217.
2009
Identification, structure-activity relationships and molecular modeling of potent triamine and piperazine opioid ligands
. 17:5583-5597.
2009
Monoquaternary pyridinium salts with modified side chain - synthesis and evaluation on model of tabun- and paraoxon-inhibited acetylcholinesterase
. 16:8218-8223.
2008
Conformation-opioid activity relationships of bicyclic guanidines from 3D similarity analysis
. 16:5932-5938.
2008
Synthesis of 5′-functionalized nucleosides::
S
-Adenosylhomocysteine analogues with the carbon-5′ and sulfur atoms replaced by a vinyl or halovinyl unit
. 16:5424-5433.
2008
S
-ribosylhomocysteine analogues with the carbon-5 and sulfur atoms replaced by a vinyl or (fluoro)vinyl unit
. 16:5090-5102.
2008
Rate enhancement of the oxidative folding of lysozyme by the use of aromatic thiol containing redox buffers
. 16:2579-2590.
2008
Monooxime reactivators of acetylcholinesterase with (
E
)-but-2-ene linker -: Preparation and reactivation of tabun- and paraoxon-inhibited acetylcholinesterase
. 15:6733-6741.
2007
Lead optimization of 7-benzyloxy 2-(4 '-pyridylmethyl)thio isoflavone aromatase inhibitors
. 13:6571-6577.
2005
Synthesis and characterization of azole isoflavone inhibitors of aromatase
. 13:4063-4070.
2005
Identification of novel small-molecule Ulex europaeus I mimetics for targeted drug delivery
. 11:4991-4997.
2003
The structural basis for kainoid selectivity at AMPA receptors revealed by low-mode docking calculations
. 11:551-559.
2003
The synthesis of peptidomimetic combinatorial libraries through successive amide alkylations
1996
Research
category
BIOCHEMISTRY & MOLECULAR BIOLOGY
Category
CHEMISTRY, MEDICINAL
Category
CHEMISTRY, ORGANIC
Category
Identifiers
International Standard Serial Number (ISSN)
0968-0896
Electronic International Standard Serial Number (EISSN)
1464-3391
Other
journal abbreviation
BIOORGAN MED CHEM