Small-Molecule Inhibitors Targeting Topoisomerase I as Novel Antituberculosis Agents Article

Sandhaus, Shayna, Annamalai, Thirunavukkarasu, Welmaker, Greg et al. (2016). Small-Molecule Inhibitors Targeting Topoisomerase I as Novel Antituberculosis Agents . ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 60(7), 4028-4036. 10.1128/AAC.00288-16

Open Access International Collaboration

cited authors

  • Sandhaus, Shayna; Annamalai, Thirunavukkarasu; Welmaker, Greg; Houghten, Richard A; Paz, Carlos; Garcia, Pamela K; Andres, Angelo; Narula, Gagandeep; Felix, Carolina Rodrigues; Geden, Sandra; Netherton, Mandy; Gupta, Rashmi; Rohde, Kyle H; Giulianotti, Marc A; Tse-Dinh, Yuk-Ching

sustainable development goals

publication date

  • July 1, 2016

published in

keywords

  • ANTIBACTERIAL COMPOUNDS
  • CLEAVAGE
  • DNA TOPOISOMERASES
  • ESCHERICHIA-COLI
  • GYRASE GENES
  • Life Sciences & Biomedicine
  • MUTATIONS
  • MYCOBACTERIUM-TUBERCULOSIS
  • Microbiology
  • Pharmacology & Pharmacy
  • SCAFFOLD RANKING
  • SYNTHETIC COMBINATORIAL LIBRARIES
  • Science & Technology
  • TN5 TRANSPOSASE

Digital Object Identifier (DOI)

publisher

  • AMER SOC MICROBIOLOGY

start page

  • 4028

end page

  • 4036

volume

  • 60

issue

  • 7