Novel selective human melanocortin-3 receptor ligands:: Use of the 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one (Aba) scaffold Article

Ballet, Steven, Mayorov, Alexander V, Cai, Minying et al. (2007). Novel selective human melanocortin-3 receptor ligands:: Use of the 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one (Aba) scaffold . BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 17(9), 2492-2498. 10.1016/j.bmcl.2007.02.020

Open Access International Collaboration

cited authors

  • Ballet, Steven; Mayorov, Alexander V; Cai, Minying; Tymecka, Dagmara; Chandler, Kevin B; Palmer, Erin S; Van Rompaey, Karolien; Misicka, Aleksandra; Tourwe, Dirk; Hruby, Victor J

sustainable development goals

authors

publication date

  • May 1, 2007

published in

keywords

  • 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-ones
  • ALPHA-MELANOTROPIN
  • ANALOGS
  • ANTAGONISTS
  • BIOLOGICAL EVALUATION
  • Chemistry
  • Chemistry, Medicinal
  • Chemistry, Organic
  • DESIGN
  • DISCOVERY
  • Life Sciences & Biomedicine
  • MINIMAL ACTIVE SEQUENCE
  • PEPTIDES
  • POTENT
  • Pharmacology & Pharmacy
  • Physical Sciences
  • SKIN BIOASSAY
  • Science & Technology
  • conformational restrictions
  • cyclic lactam analogues
  • hMC3R/hMC5R antagonists
  • human melanocortin receptors

Digital Object Identifier (DOI)

publisher

  • PERGAMON-ELSEVIER SCIENCE LTD

start page

  • 2492

end page

  • 2498

volume

  • 17

issue

  • 9