Solid-phase synthesis of 2,3,5,6-tetrahydro-1H-imidazo[1,2-a]benzo[d]- [1,3]diazepines via Pd(OAc)2/Cu(OAc)2-cocatalyzed cyclization Article

Ou, L, Shao, Z, Chen, W et al. (2011). Solid-phase synthesis of 2,3,5,6-tetrahydro-1H-imidazo[1,2-a]benzo[d]- [1,3]diazepines via Pd(OAc)2/Cu(OAc)2-cocatalyzed cyclization . SYNLETT, (15), 2259-2261. 10.1055/s-0030-1261186

cited authors

  • Ou, L; Shao, Z; Chen, W; Giulianotti, MA; Houghten, RA; Yu, Y

authors

abstract

  • An efficient approach for the solid-phase synthesis of 2,3,5,6-tetrahydro- 1H-imidazo[1,2-a]benzo[d][1,3]diazepines has been developed. It was realized by Pd(OAc)2/Cu(OAc)2-cocatalyzed intramolecular aryl guanidinylation. © Georg Thieme Verlag Stuttgart - New York.

publication date

  • August 15, 2011

published in

Digital Object Identifier (DOI)

start page

  • 2259

end page

  • 2261

issue

  • 15