Discovery of novel bacterial topoisomerase I inhibitors by use of in silico docking and in vitro assays Article

Sandhaus, Shayna, Chapagain, Prem P, Tse-Dinh, Yuk-Ching. (2018). Discovery of novel bacterial topoisomerase I inhibitors by use of in silico docking and in vitro assays . SCIENTIFIC REPORTS, 8 10.1038/s41598-018-19944-4

Open Access

keywords

  • ANTIBIOTICS
  • CLEAVAGE
  • DNA TOPOISOMERASES
  • DRUG DISCOVERY
  • ERA
  • ESCHERICHIA-COLI
  • FORCE-FIELD
  • MOLECULAR-DYNAMICS
  • Multidisciplinary Sciences
  • RESISTANCE
  • Science & Technology
  • Science & Technology - Other Topics

Digital Object Identifier (DOI)

publisher

  • NATURE PUBLISHING GROUP

volume

  • 8