Macrolactonization of peptide thioesters catalyzed by imidazole and its application in the synthesis of kahalalide B and analogues Article

Li, Y, Giulionatti, M, Houghten, RA. (2010). Macrolactonization of peptide thioesters catalyzed by imidazole and its application in the synthesis of kahalalide B and analogues . ORGANIC LETTERS, 12(10), 2250-2253. 10.1021/ol100596p

cited authors

  • Li, Y; Giulionatti, M; Houghten, RA

authors

abstract

  • The macrolactonization of peptide thioester to yield cyclic depsipeptides was developed using imidazole as a catalyst. This strategy was applied to the synthesis of kahalalide B and its analogues. © 2010 American Chemical Society.

publication date

  • May 21, 2010

published in

Digital Object Identifier (DOI)

start page

  • 2250

end page

  • 2253

volume

  • 12

issue

  • 10