Identification of an Orally Bioavailable Quinoline-Based Small-Molecule Tumor Necrosis Factor α (TNF-α) Inhibitor Featuring a Spirocyclic Scaffold Article

Sun, Zeren, Zhang, Wenbin, He, Wanyong et al. (2026). Identification of an Orally Bioavailable Quinoline-Based Small-Molecule Tumor Necrosis Factor α (TNF-α) Inhibitor Featuring a Spirocyclic Scaffold . JOURNAL OF MEDICINAL CHEMISTRY, 69(8), 8987-9008. 10.1021/acs.jmedchem.5c03457

International Collaboration

cited authors

  • Sun, Zeren; Zhang, Wenbin; He, Wanyong; Xu, Jie; Wang, Boning; He, Joshua M; Zhang, Yuchen; Chen, Pu; Luo, Yao; Gu, Jia; Gu, Hongfeng; Wei, Ping; Sun, Yanan; Yin, Chunxiang; Xing, Hanxi; Luo, Yannan; Zhang, Jing-jing; Zhu, Qihua; Zou, Yi; Xu, Yungen

sustainable development goals

authors

publication date

  • April 23, 2026

published in

keywords

  • Chemistry, Medicinal
  • Life Sciences & Biomedicine
  • Pharmacology & Pharmacy
  • RISK
  • Science & Technology

Digital Object Identifier (DOI)

publisher

  • AMER CHEMICAL SOC

start page

  • 8987

end page

  • 9008

volume

  • 69

issue

  • 8