Screening, Deconvolution and Parallel Synthesis of Trisubstituted Piperazine and Trisubstituted 2,3-diketopierazine Libraries for the Rapid Identification of Antagonists of the Nuclear Retinoic Acid Receptor-related Orphan Receptor Gamma (RORγ) Letter

Ortiz, Maria A, Piedrafita, Francisco J, Bunnell, Ashley et al. (2024). Screening, Deconvolution and Parallel Synthesis of Trisubstituted Piperazine and Trisubstituted 2,3-diketopierazine Libraries for the Rapid Identification of Antagonists of the Nuclear Retinoic Acid Receptor-related Orphan Receptor Gamma (RORγ) . 21(5), 829-835. 10.2174/1570180820666230130093524

cited authors

  • Ortiz, Maria A; Piedrafita, Francisco J; Bunnell, Ashley; Nefzi, Adel

sustainable development goals

authors

publication date

  • January 1, 2024

keywords

  • CELLS
  • Chemistry, Medicinal
  • DIFFERENTIATION
  • DISCOVERY
  • LIGANDS
  • Life Sciences & Biomedicine
  • PEPTIDES
  • POTENT
  • Pharmacology & Pharmacy
  • ROR gamma
  • SCAFFOLD RANKING
  • SOLID-PHASE SYNTHESIS
  • Science & Technology
  • antagonist
  • combinatorial chemistry
  • diketopiperazine
  • orphan receptor gamma
  • piperazine

Digital Object Identifier (DOI)

publisher

  • BENTHAM SCIENCE PUBL LTD

start page

  • 829

end page

  • 835

volume

  • 21

issue

  • 5